Category
Bedaquiline fumarate
CAS Number
2924118-10-3
Molecular Formula
C31H29BrN2O2
Molecular Weight
541.5g/mol
Synonym

6-Bromo-3-((1R,2S)-4-(dimethylamino)-2-hydroxy-2-(naphthalen-1-yl)-1-phenylbutyl)quinolin-2(1H)-one; 6-bromo-3-((1R,2S)-4-(dimethylamino)-2-hydroxy-2-(naphthalen-1-yl)-1-phenylbutyl)quinolin-2-ol; O-Desmethyl Bedaquiline

Keywords
Aromatics
Enzyme inhibitors
Pharmaceutical Standards
Fine Chemicals
Heterocycles
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O-Desmethyl Bedaquiline is a metabolite of Bedaquiline formed in the liver by the CYP3A4 enzyme. It has weaker activity against tuberculosis but can contribute to side effects like heart rhythm changes.